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ALL ABOUT DRUGS
DR ANTHONY MELVIN CRASTO Ph.D ( ICT, Mumbai) , INDIA 25Yrs Exp. in the feld of Organic Chemistry,Working for GLENMARK GENERICS at Navi Mumbai, INDIA. Serving chemists around the world. Helping them with websites on Chemistry.Million hits on google,world acclamation from industry, academia, drug authorities for websites, blogs and educational contribution, [email protected]..........+91 9323115463
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Ceftobiprole
C20H22N8O6S2
534.57
209467-52-7
(6R,7R)-7-[(2Z)-2-(5-amino-1,2,4-thiadiazol-3-yl)-2-(N-hydroxyimino)acetamido]-8-oxo-3-{[(3E,3’R)-2-oxo-[1,3′-bipyrrolidin]-3-ylidene]methyl}-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
BAL-9141
BAL-9141-000
BAL-9141000
BAL9141-000
RO 63-9141
RO-63-9141
RO-639141
ceftobiprole medocaril sodium
Ro-655788
BAL-5788-001
Molecular…
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#approvals 2024#BAL-9141#BAL-9141-000#BAL-9141000#BAL9141-000#Ceftobiprole#Ceftobiprole medocaril sodium salt#fda 2024#RO 63-9141#RO-63-9141#RO-639141#zevtera
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DANICOPAN
Danicopan
USFDA 3/29/2024, To treat extravascular hemolysis with paroxysmal nocturnal hemoglobinuria, Voydeya
C26H23BrFN7O3
580.418
1903768-17-1
(2S,4R)-1-[2-[3-acetyl-5-(2-methylpyrimidin-5-yl)indazol-1-yl]acetyl]-N-(6-bromopyridin-2-yl)-4-fluoropyrrolidine-2-carboxamide
ACH 0144471
ACH-4471
ACH0144471
ALXN 2040
ALXN-2040
ALXN2040
Danicopan, sold under the brand name Voydeya, is a…
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INAXAPLIN
INAXAPLIN, 2446816-88-0
2446816-88-0
S2SJ2RVZ6Y
UNII-S2SJ2RVZ6Y
C21H18F3N3O3
3-[5,7-difluoro-2-(4-fluorophenyl)-1H-indol-3-yl]-N-[(3S,4R)-4-hydroxy-2-oxopyrrolidin-3-yl]propanamide
Inaxaplin (VX-147) is a small-molecule apolipoprotein L1 inhibitor developed by Vertex Pharmaceuticals for APOL1-mediated kidney disease. In preliminary studies the drug has shown promise in treating people with…
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Golcadomide (CC-99282)
Golcadomide (CC-99282)
Molecular Weight535.57FormulaC28H30FN5O5CAS…
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Oditrasertib,
Obeldesivir,
2647441-36-7
361.35 g/mol
C16H19N5O5
[(2R,3S,4R,5R)-5-(4-aminopyrrolo[2,1-f][1,2,4]triazin-7-yl)-5-cyano-3,4-dihydroxyoxolan-2-yl]methyl 2-methylpropanoate
Q55KCM7PXB; ATV006; UNII-Q55KCM7PXB
Obeldesivir (GS-5245, ATV006) is an isobutyric ester prodrug of GS-441524 made by Gilead Sciences that is currently in Phase III trials for the outpatient treatment of COVID-19 in high…
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ORZILOBEN
ORZILOBEN,
CAS 1555822-28-0
2-methyl-3-(pentyloxy)benzoic acid
Molecular Weight222.28FormulaC13H18O3
Orziloben is a medium chain fatty acid (MCFA) analogue[1].
Patent
WO2020074964
https://patentscope.wipo.int/search/en/detail.jsf?docId=WO2020074964&_cid=P12-LQYZJX-26404-1
The rising global epidemic of obesity and its comorbidities, e.g., type 2 diabetes mellitus and hyperlipidemia, is…
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Sotuletinib HCl
Sotuletinib HCl
CAS: 2222138-31-8 (HCl)Chemical Formula: C20H23ClN4O3S
Molecular Weight: 434.939
7W3V82OQ0P
Synonym: Sotuletinib HCl; Sotuletinib hydrochloride, Sotuletinib monohydrochloride, BLZ945; BLZ 945; BLZ-945;
IUPAC/Chemical Name: 4-((2-(((1R,2R)-2-hydroxycyclohexyl)amino)benzo[d]thiazol-6-yl)oxy)-N-methylpicolinamide hydrochloride
2-PYRIDINECARBOXAMIDE,…
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Eplontersen
Eplontersen
AKCEA-TTR-LRx
ION-682884 FREE ACID
ISIS-682884 FREE ACID
UNII0GRZ0F5XJ6
CAS…
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Eplontersen
Eplontersen
AKCEA-TTR-LRx
ION-682884 FREE ACID
ISIS-682884 FREE ACID
UNII0GRZ0F5XJ6
CAS…
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Iptacopan
Iptacopan
1644670-37-0
422.525, C25H30N2O4
4-((2S,4S)-4-ethoxy-1-((5-methoxy-7-methyl-1H-indol-4-yl)methyl)piperidin-2-yl) benzoic acid
BENZOIC ACID, 4-((2S,4S)-4-ETHOXY-1-((5-METHOXY-7-METHYL-1H-INDOL-4-YL)METHYL)-2-PIPERIDINYL)-
Iptacopan
LNP 023
LNP-023
LNP023
NVP-LNP023
NVP-LNP023-NX
fda approved, To treat paroxysmal nocturnal hemoglobinuria, 12/5/2023, Fabhalta ‘
Iptacopan is a…
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#12/5/2023#2023#APPROVALS#Fabhalta#FDA 2023#Iptacopan#LNP 023#LNP-023#LNP023#NVP-LNP023#NVP-LNP023-NX#paroxysmal nocturnal hemoglobinuria
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CAREBASTINE
CAREBASTINE
Molecular Weight499.64AppearanceSolidFormulaC32H37NO4CAS No.90729-42-3
Carebastine is the active metabolite of Ebastine. Carebastine is a histamine H1 receptor antagonist. Carebastine inhibits VEGF-induced HUVEC and HPAEC proliferation, migration and angiogenesis in a dose-dependent manner. Carebastine suppresses the expression of macrophage migration inhibitory factor.
Carebastine…
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VODOBATINIB
VODOBATINIB
1388803-90-4
Molecular Weight453.92AppearanceSolidFormulaC27H20ClN3O2
SCO-088
K0706
K-0706
2-chloro-6-methyl-N‘-[4-methyl-3-(2-quinolin-3-ylethynyl)benzoyl]benzohydrazide
Vodobatinib (K0706) is a potent, third generation and orally active Bcr-Abl1 tyrosine kinase inhibitor with an IC50 of 7 nM. Vodobatinib exhibits activity against most BCR-ABL1 point mutants, and has no…
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Etrasimod
Etrasimod
APD334
C26H26F3NO3
457.493
1206123-37-62-[(3R)-7-{[4-cyclopentyl-3-(trifluoromethyl)phenyl]methoxy}-1H,2H,3H,4H-cyclopenta[b]indol-3-yl]acetic acid
Etrasimod arginineMXE5EMA09L1206123-97-8GVPVVOSNDUAUKM-BPGOJFKZSA-N
Name: Etrasimod arginineCAS#: 1206123-97-8 (arginine)Chemical Formula: C32H40F3N5O5Exact Mass: 631.30Molecular Weight: 631.700
FDA APPROVED, To treat moderately to…
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Motixafortide
Motixafortide
4F-benzoyl-TN-14003
BKT-140
BKT140
BL-8040
Protein Chemical FormulaC97H144FN33O19S2
Protein Average Weight2159.6 Da
UNIIDA9G065962CAS number664334-36-5>Motixafortide sequence RRXCYXKKPYRXCR
Motixafortide acetate 2639893-42-6GMUZYOKQKWMETH-AQDOTSTFSA-N
fda approved,9/8/2023,
Aphexda
мотиксафортид[Russian]
موتيكسافورتيد[Arabic]
莫替福肽[Chinese]
Motixafortide is a peptide…
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#4F-benzoyl-TN-14003#Aphexda#APPROVALS 2023#BKT-140#BKT140#BL 8040#da 2023#мотиксафортид#莫替福肽#Motixafortide#موتيكسافورتيد
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EIDD-2173, ATI-2173
EIDD-2173; also known as ATI-2173
Hepatitis B virus (HBV) is an infectious disease that targets the liver resulting in either an acute infection, with symptoms arising in 45 to 160 days, or a chronic infection, which 350 million people worldwide are affected by. Estimates indicate that 600,000 deaths occur each year as a result of consequences related to HBV infection. HBV possesses a 3.2- kb…
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